Acetyl-Calpastatin (184-210) (human)

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断

Selective calpain inhibitor. Strongly inhibits calpain I (Ki = 0.2 nM) and II but does not inhibit papain, trypsin and cathepsin L (Ki = 6 μM). Increases secretion of amyoid β-protein (Aβ) 42, Aβ40 and Aβ42 ratio.

Selective calpain inhibitor. Strongly inhibits calpain I (Ki = 0.2 nM) and II but does not inhibit papain, trypsin and cathepsin L (Ki = 6 μM). Increases secretion of amyoid β-protein (Aβ) 42, Aβ40 and Aβ42 ratio.

Acetyl-Calpastatin(184-210)(human) (peptide 1; 12.5-100 μM) inhibits calpains in LCLC 103H cells with an IC50 of 27 μM.

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Proteasome/Ubiquitin

Proteasome

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123714-50-1

3177.65

C142H230N36O44S

>98% (HPLC)

water:5 mg/mL

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(-20℃)

With Ice Pack

≥ 2 years